Selection of our most important completed research projects

This project studies the key step in the biosynthesis of phloridzin, which is the prevalent polyphenolic compound in apple. Phloridzin represents more than 90% of the soluble phenolic compounds in apple leaves. The presence of such high amounts of phloridzin makes apple unique since other species accumulate only very low amounts and many closely related species like pear are not able to form phloretin or its glucosylated relative phloridzin. The last decade has seen an explosion of research on the beneficial effects of phloretin and phloridzin for human health but the physiological relevance for apple is still unclear. A possible involvement in disease resistance is discussed. Previously we have shown with apple leaf extracts that phloridzin formation is based on three biosynthetic steps: (1) the formation of dihydro-p-coumaroyl-CoA from p-coumaroyl-CoA by a dehydrogenase, (2) further formation of phloretin by the common chalcone synthase and (3) the glucosylation of phloretin in position 2’. Whereas the last two steps were already intensively studied, the knowledge of the first step is limited. The enzyme is crucial, because it seems to be the key point making the phloridzin-hoarding apple unique in comparison to other plants. In our previous FWF project (P25399-B16) we successfully completed a challenging purification process and were able to purify for the first time a candidate enzyme from apple leaves, which exhibits strong enzyme activity with p-coumaroyl-CoA to form dihydro-p-coumaroyl-CoA. The planned follow-up project will now target the detailed characterization of this important enzyme from apple leaves for the first time. Structural studies will resolve the enzymatic mechanism, such as protein crystallization and effects of substrates, inhibitors/effectors or other factors. The DNA sequence of the dehydrogenase will be isolated from apple and transferred into bacteria to produce large amounts of the enzyme for detailed characterization. It will be tested, in which tissue and developmental stage the dehydrogenase gene is switched on or off.  Functional activity of the gene products will be tested with genetically modified plants where phloretin formation will be enabled by the dehydrogenase in thale cress (Arabidopsis) or disabled in apple. Comparison of the DNA and protein sequence of the dehydrogenase from different plant species will give insight to structure-activity relationship of the enzyme on the molecular level. The project members consist of three teams which provide complementary know-how and resources: One of the Austrian teams offers knowledge in phloridzin biosynthesis, molecular biology and enzymatic evaluation, the other Austrian team has profound experience in protein characterization and crystallisation, whereas the German team provides the infrastructure and long-term experience in the creation of transgenic plants. An external team from New Zealand, which is funded by own sources will additionally contribute its know-how on pear transformation.

Funding: FWF - Austrian Science Fund and DFG - Deutsche Forschungsgemeinschaft

Project number: I 4296

Duration: 01.05.2020 – 30.04.2024

Contact: Senior Scientist Dipl.-Ing. Dr.rer.nat. Christian Haselmair-Gosch

PUBLICATIONS

Cebulj A, Mikulic-Petkovsek M, Lucaciu C, Veberic R, Marinovic S, Kolarek M, Hutabarat OS, Faramarzi S, Rattei T, Molitor C, Hudina M, Haselmair-Gosch C, Halbwirth H, Slatnar A. (2021). Alteration of the phenylpropanoid pathway by watercore disorder in apple (Malus x domestica). Scientia Horticulturae, https://doi.org/10.1016/j.scienta.2021.110438, opens an external URL in a new window

Weissensteiner J, Molitor C, Marinovic S, Führer L, Waqas Hassan S, Hutabarat OS, Spornberger A, Stich K, Hausjell J, Spadiut O, Haselmair-Gosch C, Halbwirth H. (2021). Molecular and Enzymatic Characterization of Flavonoid 3'-Hydroxylase of Malus × domestica. Plants (Basel, Switzerland), 10(9), https://doi.org/10.3390/plants10091956, opens an external URL in a new window

Schröpfer S., Molitor C., Haselmair-Gosch C., Flachowsky H., Stich K., Halbwirth H. (2022). XXXI International Horticultural Congress (IHC2022): International Symposium on Breeding and Effective Use of Biotechnology and Molecular Tools in Horticultural Crops. 31st International Horticultural Congress: International Symposium on Breeding and Effective Use of Biotechnology and Molecular Tools in Horticultural Crops.

Schröpfer S., Molitor C., Haselmair-Gosch C., Flachowsky H., Stich K., Halbwirth H. (2023). Polyphenols Communications e-vol. 2. The International Conference on Polyphenols (ICP).

Schröpfer S., Molitor C., Böttcher C., Haselmair-Gosch C., Flachowsky H., Halbwirth H. (2023). Validation of a candidate gene involved in the biosynthesis of phloridzin in apple by heterologous expression in Arabidopsis thaliana. XVI Eucarpia Symposium on Fruit Breeding and Genetics.

Kornpointner C., Miksovsky P., Rabeeah I.A., Murray H., Goessinger M., Haselmair-Gosch C., Stich K., Bica-Schroeder K., Halbwirth H. (2023). Polyphenols Communications e-vol. 2. The International Conference on Polyphenols (ICP).

Kniely J. (2021). Molecularbiological and biochemical investigations on the dihydrochalcone biosynthesis in apple leaves. Bachelor thesis

Metzgen M. (2020). Herstellung und Charakterisierung von rekombinanten Cytochrom-P450-abhängigen Proteinen aus Angelonien und Apfel. Bachelorarbeit

Schmidt-Gruber V. (2024). Hinter die Schale geschaut: Verteilung von Phloridzin in verschiedenen Apfelteilen und Untersuchungen zu seiner antioxidativen Wirkung. Bachelorarbeit

Schöpf M. (2022). Untersuchungen zur Reaktion der Chalkonsynthase. Diplomarbeit

This project studies the key step in the biosynthesis of phloridzin, which is the prevalent polyphenolic compound in apple. Phloridzin represents more than 90% of the soluble phenolic compounds in apple leaves. The presence of such high amounts of phloridzin makes apple unique since other species accumulate only very low amounts and many closely related species like pear are not able to form phloretin or its glucosylated relative phloridzin. The last decade has seen an explosion of research on the beneficial effects of phloretin and phloridzin for human health but the physiological relevance for apple is still unclear. A possible involvement in disease resistance is discussed. Previously we have shown with apple leaf extracts that phloridzin formation is based on three biosynthetic steps: (1) the formation of dihydro-p-coumaroyl-CoA from p-coumaroyl-CoA by a dehydrogenase, (2) further formation of phloretin by the common chalcone synthase and (3) the glucosylation of phloretin in position 2’. Whereas the last two steps were already intensively studied, the knowledge of the first step is limited. The enzyme is crucial, because it seems to be the key point making the phloridzin-hoarding apple unique in comparison to other plants. In our previous FWF project (P25399-B16) we successfully completed a challenging purification process and were able to purify for the first time a candidate enzyme from apple leaves, which exhibits strong enzyme activity with p-coumaroyl-CoA to form dihydro-p-coumaroyl-CoA. The planned follow-up project will now target the detailed characterization of this important enzyme from apple leaves for the first time. Structural studies will resolve the enzymatic mechanism, such as protein crystallization and effects of substrates, inhibitors/effectors or other factors. The DNA sequence of the dehydrogenase will be isolated from apple and transferred into bacteria to produce large amounts of the enzyme for detailed characterization. It will be tested, in which tissue and developmental stage the dehydrogenase gene is switched on or off.  Functional activity of the gene products will be tested with genetically modified plants where phloretin formation will be enabled by the dehydrogenase in thale cress (Arabidopsis) or disabled in apple. Comparison of the DNA and protein sequence of the dehydrogenase from different plant species will give insight to structure-activity relationship of the enzyme on the molecular level. The project members consist of three teams which provide complementary know-how and resources: One of the Austrian teams offers knowledge in phloridzin biosynthesis, molecular biology and enzymatic evaluation, the other Austrian team has profound experience in protein characterization and crystallisation, whereas the German team provides the infrastructure and long-term experience in the creation of transgenic plants. An external team from New Zealand, which is funded by own sources will additionally contribute its know-how on pear transformation.

Funding: FWF - Austrian Science Fund

Project number: P 32901

Duration: 01.01.2020 – 31.12.2023

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth

PUBLICATIONS

Walliser, Benjamin, Silvija Marinovic, Christoph Kornpointner, Christopher Schlosser, Mustafa Abouelnasr, Olly Sanny Hutabarat, Christian Haselmair-Gosch, Christian Molitor, Karl Stich, and Heidi Halbwirth. "The (Bio) chemical Base of Flower Colour in Bidens ferulifolia." Plants 11, no. 10 (2022): 1289. https://doi.org/10.3390/plants11101289, opens an external URL in a new window

Weissensteiner, Julia, Christian Molitor, Silvija Marinovic, Lisa Führer, Syed Waqas Hassan, Olly Sanny Hutabarat, Andreas Spornberger, Karl Stich, Johanna Hausjell, Oliver Spadiut, Christian Haselmair-Gosch, and Heidi Halbwirth "Molecular and Enzymatic Characterization of Flavonoid 3′-Hydroxylase of Malus × domestica." Plants 10, no. 9 (2021): 1956.   https://doi.org/10.3390/plants10091956, opens an external URL in a new window

Walliser, Benjamin, Calin Rares Lucaciu, Christian Molitor, Silvija Marinovic, Daria Agata Nitarska, Didem Aktaş, Thomas Rattei, Ioannis Kampatsikas, Karl Stich, Christian Haselmair-Gosch and Heidi Halbwirth "Dahlia variabilis cultivar ‘Seattle’ as a model plant for anthochlor biosynthesis." Plant Physiology and Biochemistry 159 (2021): 193-201. https://doi.org/10.1016/j.plaphy.2020.12.016, opens an external URL in a new window

Nitarska, D., Boehm, R., Debener, T., Lucaciu, R. C., & Halbwirth, H. (2021). First genome edited poinsettias: targeted mutagenesis of flavonoid 3′-hydroxylase using CRISPR/Cas9 results in a colour shift. Plant Cell, Tissue and Organ Culture (PCTOC), 1-12. https://doi.org/10.1007/s11240-021-02103-5, opens an external URL in a new window

Cebulj, Anka, Maja Mikulic-Petkovsek, Calin Rares Lucaciu, Robert Veberic, Silvija Marinovic, Martina Kolarek, Olly Sanny Hutabarat, Shadab Faramarzi, Thomas Rattei, Christian Molitor, Metka Hudina, Christian Haselmair-Gosch, Heidi Halbwirth, and Ana Slatnar "Alteration of the phenylpropanoid pathway by watercore disorder in apple (Malus x domestica)." Scientia Horticulturae 289 (2021): 110438, https://doi.org/10.1016/j.scienta.2021.110438, opens an external URL in a new window

Hausjell, Johanna, Julia Weissensteiner, Christian Molitor, Karin Schlangen, Oliver Spadiut, and Heidi Halbwirth. "First purified recombinant CYP75B including transmembrane helix with unexpected high substrate specificity to (2R)-naringenin." Scientific Reports 12, no. 1 (2022): 1-13. DOI: https://doi.org/10.1038/s41598-022-11556-3, opens an external URL in a new window

 

Funding: WWTF Vienna Science and Technology Fund

Project number: ESR17-027

Duration: 01.03.2018 – 28.02.2023

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth

Funding: FWF - Austrian Science Fund

Project number: I 2919

Duration: 2017 - 2021

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth

Funding: European Commission, Horizon2020

Project number: 675657

Duration: 2016 - 2020

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth

Funding: FWF - Austrian Science Fund

Project number: P 29552

Duration: 2016 - 2019

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth

Funding: FWF - Austrian Science Fund

Project number: P 28795

Duration: 2016 - 2019

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth

Funding: FWF - Austrian Science Fund

Project number: P 28134

Duration: 2015 - 2020

Contact: Senior Scientist Dipl.-Ing. Dr.rer.nat. Christian Haselmair-Gosch

Funding: FWF - Austrian Science Fund

Project number: P 26468

Duration: 2014 - 2018

Contact: Ao.Univ.-Prof.i.R. Dipl.-Ing. Dr.nat.techn. Karl Stich

Funding: FWF - Austrian Science Fund

Project number: P 25399

Duration: 2013 - 2018

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth

Funding: FWF - Austrian Science Fund

Project number: P 24331

Duration: 2012 - 2015

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth

Funding: European Commission (Euphresco)

Project number: 100867

Duration: 2012 - 2014

Contact: Ao.Univ.-Prof.i.R. Dipl.-Ing. Dr.nat.techn. Karl Stich

Funding: Austrian Federal Ministry for Economy, Family and Youth (PRIZE 2010)

Project number: Z100355

Duration: 2012 - 2014

Contact: Ao.Univ.-Prof.i.R. Dipl.-Ing. Dr.nat.techn. Karl Stich

Funding: Austrian Federal Ministry of Agriculture, Forestry, Environment and Water Management

Project number: 100404

Duration: 2008 - 2011

Contact: Ao.Univ.-Prof.i.R. Dipl.-Ing. Dr.nat.techn. Karl Stich

Funding: Gesellschaft zur Förderung von Pflanzenforschung

Duration: 2008

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth

Funding: FWF - Austrian Science Fund

Project number: V18-B03

Duration: 2006 - 2011

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth

Funding: European Commission

Project number:

Duration: 2006 - 2010

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth

Funding: European Science Foundation

Project number: COST Action 864

Duration: 2006 - 2010

Contact: Ao.Univ.-Prof.i.R. Dipl.-Ing. Dr.nat.techn. Karl Stich

Funding: FWF - Austrian Science Fund

Project number: P 17629

Duration: 2004 - 2006

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth

Funding: Hochschuljubiläumsstiftung der Stadt Wien

Project number:

Duration: 2002 - 2004

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth

Funding: European Commission

Project number: QLK5-CT-1999-01583

Duration: 2000 – 2003

Contact: Ao.Univ.-Prof.i.R. Dipl.-Ing. Dr.nat.techn. Karl Stich

Funding: FWF - Austrian Science Fund

Project number: P 13020

Duration: 1999 - 2000

Contact: Ao.Univ.-Prof.i.R. Dipl.-Ing. Dr.nat.techn. Karl Stich

Funding: Jubiläumsfonds der Österreichischen Nationalbank

Project number:

Duration: 1999 - 2000

Contact: Associate Prof. Dipl.-Ing. Dr.in techn. Heidi Halbwirth